Bařinka, Cyril: шукати на сайті Z-Library

Journal of Neurochemistry

Рік:

2004

Мова:

english

Файл:

PDF, 181 KB

english, 2004

Biochemical characterization of human glutamate carboxypeptidase III

Klára Hlouchová, Cyril Bařinka, Vojtěch Klusák, Pavel Šácha, Petra Mlčochová, Pavel Majer, Lubomír Rulíšek, Jan Konvalinka

Журнал:

Рік:

2007

Мова:

english

Файл:

PDF, 1.21 MB

english, 2007

Mapping of the active site of glutamate carboxypeptidase II by site-directed mutagenesis

Petra Mlčochová, Anna Plechanovová, Cyril Bařinka, Daruka Mahadevan, Jose W. Saldanha, Lubomír Rulíšek, Jan Konvalinka

Журнал:

Klara Hlouchova, Cyril Barinka, Jan Konvalinka, Jacek Lubkowski

Рік:

2007

Мова:

english

Файл:

PDF, 866 KB

english, 2007

Structural insight into the evolutionary and pharmacologic homology of glutamate carboxypeptidases II and III

Журнал:

Archives of Biochemistry and Biophysics

Рік:

2009

Мова:

english

Файл:

PDF, 916 KB

english, 2009

Structure of glutamate carboxypeptidase II, a drug target in neuronal damage and prostate cancer

Mesters, Jeroen R, Barinka, Cyril, Li, Weixing, Tsukamoto, Takashi, Majer, Pavel, Slusher, Barbara S, Konvalinka, Jan, Hilgenfeld, Rolf

Журнал:

The EMBO Journal

Рік:

2006

Мова:

english

Файл:

PDF, 366 KB

english, 2006

A Picomolar Inhibitor of Resistant Strains of Human Immunodeficiency Virus Protease Identified by a Combinatorial Approach

Markéta Rinnová, Martin Hradilek, Cyril Bařinka, Jan Weber, Milan Souček, Jiřı́ Vondrášek, Thomas Klimkait, Jan Konvalinka

Журнал:

Рік:

2000

Мова:

english

Файл:

PDF, 684 KB

english, 2000

Structural Basis of Interaction between Urokinase-type Plasminogen Activator and its Receptor

Cyril Barinka, Graham Parry, Jennifer Callahan, David E. Shaw, Alice Kuo, Khalil Bdeir, Douglas B. Cines, Andrew Mazar, Jacek Lubkowski

Журнал:

Journal of Molecular Biology

Рік:

2006

Мова:

english

Файл:

PDF, 952 KB

english, 2006

Structural Basis of Interactions between Human Glutamate Carboxypeptidase II and Its Substrate Analogs

Cyril Barinka, Klara Hlouchova, Miroslava Rovenska, Pavel Majer, Miroslawa Dauter, Niyada Hin, Yao-Sen Ko, Takashi Tsukamoto, Barbara S. Slusher, Jan Konvalinka, Jacek Lubkowski

Журнал:

Journal of Molecular Biology

Рік:

2008

Мова:

english

Файл:

PDF, 1.31 MB

english, 2008

Resonance Assignment and Three-Dimensional Structure Determination of a Human α-Defensin, HNP-1, by Solid-State NMR

Yuan Zhang, Tim Doherty, Jing Li, Wuyuan Lu, Cyril Barinka, Jacek Lubkowski, Mei Hong

Журнал:

Journal of Molecular Biology

Рік:

2010

Мова:

english

Файл:

PDF, 2.24 MB

english, 2010

Mouse brain serine racemase catalyzes specific elimination of L-serine to pyruvate

Kvido Střı́šovský, Jana Jirásková, Cyril Bařinka, Pavel Majer, Camilo Rojas, Barbara S Slusher, Jan Konvalinka

Журнал:

FEBS Letters

Рік:

2003

Мова:

english

Файл:

PDF, 141 KB

english, 2003

Identification of the N-glycosylation sites on glutamate carboxypeptidase II necessary for proteolytic activity

Cyril Barinka, Pavel Šácha, Jan Sklenář, Petr Man, Karel Bezouška, Barbara S. Slusher, Jan Konvalinka

Журнал:

Protein Science

Рік:

2004

Мова:

english

Файл:

PDF, 154 KB

english, 2004

Interactions between Human Glutamate Carboxypeptidase II and Urea-Based Inhibitors: Structural Characterization †

Barinka, Cyril, Byun, Youngjoo, Dusich, Crystal L., Banerjee, Sangeeta R., Chen, Ying, Castanares, Mark, Kozikowski, Alan P., Mease, Ronnie C., Pomper, Martin G., Lubkowski, Jacek

Журнал:

Bioorganic & Medicinal Chemistry Letters

Рік:

2008

Мова:

english

Файл:

PDF, 1.22 MB

english, 2008

Structural characterization of P1′-diversified urea-based inhibitors of glutamate carboxypeptidase II

Pavlicek, Jiri, Ptacek, Jakub, Cerny, Jiri, Byun, Youngjoo, Skultetyova, Lubica, Pomper, Martin G., Lubkowski, Jacek, Barinka, Cyril

Журнал:

Рік:

2014

Мова:

english

Файл:

PDF, 1.31 MB

english, 2014

Structural Insight into the Pharmacophore Pocket of Human Glutamate Carboxypeptidase II ⊥

Bařinka, Cyril, Rovenská, Miroslava, Mlčochová, Petra, Hlouchová, Klára, Plechanovová, Anna, Majer, Pavel, Tsukamoto, Takashi, Slusher, Barbara S., Konvalinka, Jan, Lubkowski, Jacek

Журнал:

Zhang, Andrew X., Murelli, Ryan P., Barinka, Cyril, Michel, Julien, Cocleaza, Alexandra, Jorgensen, William L., Lubkowski, Jacek, Spiegel, David A.

Рік:

2007

Мова:

english

Файл:

PDF, 292 KB

english, 2007

A Remote Arene-Binding Site on Prostate Specific Membrane Antigen Revealed by Antibody-Recruiting Small Molecules

Журнал:

Journal of the American Chemical Society

Рік:

2010

Мова:

english

Файл:

PDF, 3.36 MB

english, 2010

Homology modeling and SAR analysis of Schistosoma japonicum cathepsin D (SjCD) with statin inhibitors identify a unique active site steric barrier with potential for the design of specific inhibitors

Caffrey, Conor R., Placha, Lenka, Barinka, Cyril, Hradilek, Martin, Dostál, Jiří, Sajid, Mohammed, McKerrow, James H., Majer, Pavel, Konvalinka, Jan, Vondrášek, Jiří

Журнал:

Biological Chemistry

Рік:

2005

Мова:

english

Файл:

PDF, 351 KB

english, 2005

Structural and Biochemical Characterization of a Novel Aminopeptidase from Human Intestine

Tykvart, Jan, Bařinka, Cyril, Svoboda, Michal, Navrátil, Václav, Souček, Radko, Hubálek, Martin, Hradilek, Martin, Šácha, Pavel, Lubkowski, Jacek, Konvalinka, Jan

Журнал:

Journal of Biological Chemistry

Рік:

2015

Мова:

english

Файл:

PDF, 5.76 MB

english, 2015

A high-affinity [18F]-labeled phosphoramidate peptidomimetic PSMA-targeted inhibitor for PET imaging of prostate cancer

Ganguly, Tanushree, Dannoon, Shorouk, Hopkins, Mark R., Murphy, Stephanie, Cahaya, Hendry, Blecha, Joseph E., Jivan, Salma, Drake, Christopher R., Barinka, Cyril, Jones, Ella F., VanBrocklin, Henry F.

Журнал:

Nuclear Medicine and Biology

Рік:

2015

Мова:

english

Файл:

PDF, 457 KB

english, 2015

Carborane-containing urea-based inhibitors of glutamate carboxypeptidase II: Synthesis and structural characterization

Youn, Sihyun, Kim, Kyung Im, Ptacek, Jakub, Ok, Kiwon, Novakova, Zora, Kim, YunHye, Koo, JaeHyung, Barinka, Cyril, Byun, Youngjoo

Журнал:

Bioorganic & Medicinal Chemistry Letters

Рік:

2015

Мова:

english

Файл:

PDF, 1014 KB

english, 2015

Selection and characterization of Anticalins targeting human prostate-specific membrane antigen (PSMA)

Barinka, Cyril, Ptacek, Jakub, Richter, Antonia, Novakova, Zora, Morath, Volker, Skerra, Arne

Журнал:

Protein Engineering Design and Selection

Рік:

2016

Мова:

english

Файл:

PDF, 939 KB

english, 2016

Design of composite inhibitors targeting glutamate carboxypeptidase II: the importance of effector functionalities

Novakova, Zora, Cerny, Jiri, Choy, Cindy J., Nedrow, Jessie R., Choi, Joeseph K., Lubkowski, Jacek, Berkman, Clifford E., Barinka, Cyril

Журнал:

Nováková, Zora, Foss, Catherine A., Copeland, Benjamin T., Morath, Volker, Baranová, Petra, Havlínová, Barbora, Skerra, Arne, Pomper, Martin G., Barinka, Cyril

Рік:

2016

Мова:

english

Файл:

PDF, 1.51 MB

english, 2016

Calcium-Driven Folding of RTX Domain β-Rolls Ratchets Translocation of RTX Proteins through Type I Secretion Ducts

Bumba, Ladislav, Masin, Jiri, Macek, Pavel, Wald, Tomas, Motlova, Lucia, Bibova, Ilona, Klimova, Nela, Bednarova, Lucie, Veverka, Vaclav, Kachala, Michael, Svergun, Dmitri I., Barinka, Cyril, Sebo, Pe

Журнал:

Molecular Cell

Рік:

2016

Мова:

english

Файл:

PDF, 5.32 MB

english, 2016

Novel Monoclonal Antibodies Recognizing Human Prostate-Specific Membrane Antigen (PSMA) as Research and Theranostic Tools

Журнал:

The Prostate

Рік:

2017

Мова:

english

Файл:

PDF, 5.69 MB

english, 2017

Design and Synthesis of Mercaptoacetamides as Potent, Selective, and Brain Permeable Histone Deacetylase 6 Inhibitors

Lv, Wei, Zhang, Guangming, Barinka, Cyril, Eubanks, James H., Kozikowski, Alan P.

Журнал:

Рік:

2017

Мова:

english

Файл:

PDF, 575 KB

english, 2017

Discovery of a para-acetoxy-benzyl ester prodrug of a hydroxamate-based Glutamate Carboxypeptidase II inhibitor as oral therapy for neuropathic pain

Rais, Rana, Vávra, Jan, Tichý, Tomáš, Dash, Ranjeet P., Gadiano, Alexandra J., Tenora, Lukas, Monincova, Lenka, Barinka, Cyril, Alt, Jesse, Zimmermann, Sarah C., Slusher, C. Ethan, Wu, Ying, Wozniak,

Журнал:

Kopka, Klaus, Benešová, Martina, Bařinka, Cyril, Haberkorn, Uwe, Babich, John

Рік:

2017

Мова:

english

Файл:

PDF, 555 KB

english, 2017

Glu-Ureido–Based Inhibitors of Prostate-Specific Membrane Antigen: Lessons Learned During the Development of a Novel Class of Low-Molecular-Weight Theranostic Radiotracers

Журнал:

Journal of Nuclear Medicine

Рік:

2017

Мова:

english

Файл:

PDF, 1.42 MB

english, 2017

Synthesis and Pharmacological Evaluation of Selective Histone Deacetylase 6 Inhibitors in Melanoma Models

Tavares, Mauricio Temotheo, Shen, Sida, Knox, Tessa, Hadley, Melissa, Kutil, Zsofia, Barinka, Cyril, Villagra, Alejandro, Kozikowski, Alan P.

Журнал:

Ptacek, Jakub, Nedvedova, Jana, Navratil, Michal, Havlinova, Barbora, Konvalinka, Jan, Barinka, Cyril

Рік:

2017

Мова:

english

Файл:

PDF, 1.61 MB

english, 2017

Histone deacetylase 11 is a fatty-acid deacylase

Kutil, Zsofia, Novakova, Zora, Meleshin, Marat, Mikesova, Jana, Schutkowski, Mike, Barinka, Cyril

Журнал:

ACS Chemical Biology

Рік:

2018

Мова:

english

Файл:

PDF, 1.99 MB

english, 2018

The calcium-binding site of human glutamate carboxypeptidase II is critical for dimerization, thermal stability and enzymatic activity

Журнал:

Protein Science

Рік:

2018

Мова:

english

Файл:

PDF, 1.32 MB

english, 2018

Evaluation of 111 In-DOTA-5D3, a Surrogate SPECT Imaging Agent for Radioimmunotherapy of Prostate-Specific Membrane Antigen

Ray Banerejee, Sangeeta, Kumar, Vivek, Lisok, Ala, Plyku, Donika, Nováková, Zora, Wharram, Bryan, Brummet, Mary, Barinka, Cyril, Hobbs, Robert F, Pomper, Martin G.

Журнал:

Journal of Nuclear Medicine

Рік:

2018

Мова:

english

Файл:

PDF, 816 KB

english, 2018

2-Aminoadipic Acid-C(O)-Glutamate Based Prostate-Specific Membrane Antigen Ligands for Potential Use as Theranostics

Nakajima, Ryo, Novakova, Zora, Tueckmantel, Werner, Motlova, Lucia, Barinka, Cyril, Kozikowski, Alan P.

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2018

Мова:

english

Файл:

PDF, 2.56 MB

english, 2018

Structural and computational basis for potent inhibition of glutamate carboxypeptidase II by carbamate-based inhibitors

Barinka, Cyril, Novakova, Zora, Hin, Niyada, Bím, Daniel, V Ferraris, Dana, Duvall, Bridget, Kabarriti, Gabriel, Tsukamoto, Reiji, Budesinsky, Milos, Motlova, Lucia, Rojas, Camilo, Slusher, Barbara S.

Журнал:

Рік:

2018

Мова:

english

Файл:

PDF, 1.23 MB

english, 2018

Molecular Basis for the Selective Inhibition of Histone Deacetylase 6 by a Mercaptoacetamide Inhibitor

Porter, Nicholas J., Shen, Sida, Barinka, Cyril, Kozikowski, Alan P., Christianson, David W.

Журнал:

Рік:

2018

Мова:

english

Файл:

PDF, 2.95 MB

english, 2018

Development of Multi-Functional Histone Deacetylase 6 Degraders with Potent Anti-Myeloma Activity

Wu, Hao, Yang, Ka, Zhang, Zhongrui, Leisten, Eric, LI, ZIYUAN, Xie, Haibo, Liu, Jin, Smith, Kerry A., Novakova, Zora, Barinka, Cyril, Tang, Weiping

Журнал:

Рік:

2019

Мова:

english

Файл:

PDF, 1.30 MB

english, 2019

Development of Multi-Functional Histone Deacetylase 6 Degraders with Potent Anti-Myeloma Activity

Wu, Hao, Yang, Ka, Zhang, Zhongrui, Leisten, Eric, LI, ZIYUAN, Xie, Haibo, Liu, Jin, Smith, Kerry A., Novakova, Zora, Barinka, Cyril, Tang, Weiping

Журнал:

Рік:

2019

Файл:

PDF, 1.30 MB

2019

Discovery of a New Isoxazole-3-hydroxamate Based Histone Deacetylase 6 Inhibitor SS-208 with Anti-tumor Activity in Syngeneic Melanoma Mouse Models

Shen, Sida, Hadley, Melissa, Ustinova, Kseniya, Pavlíček, Jiří, Knox, Tessa, Noonepalle, Satish, Tavares, Mauricio Temotheo, Zimprich, Chad A., Zhang, GuiPing, Robers, Matthew B., Barinka, Cyril, KOZI

Журнал:

Hapuarachchige, Sudath, Huang, Colin T., Donnelly, Madeline C., Bařinka, Cyril, Lupold, Shawn E., Pomper, Martin G., Artemov, Dmitri

Рік:

2019

Мова:

english

Файл:

PDF, 1.11 MB

english, 2019

One-Atom-Substitution Enables Direct and Continuous Monitoring of Histone Deacylase Activity

Zessin, Matthes, Kutil, Zsófia, Meleshin, Marat, Novakova, Zora, Ghazy, Ehab, Kalbas, Diana, Marek, Martin, Romier, Christophe, Sippl, Wolfgang, Bařinka, Cyril, Schutkowski, Mike

Журнал:

Biochemistry

Рік:

2019

Мова:

english

Файл:

PDF, 1.89 MB

english, 2019

One-Atom-Substitution Enables Direct and Continuous Monitoring of Histone Deacylase Activity

Zessin, Matthes, Kutil, Zsófia, Meleshin, Marat, Novakova, Zora, Ghazy, Ehab, Kalbas, Diana, Marek, Martin, Romier, Christophe, Sippl, Wolfgang, Bařinka, Cyril, Schutkowski, Mike

Журнал:

Biochemistry

Рік:

2019

Файл:

PDF, 1.89 MB

2019

Cellular Delivery of Bioorthogonal Pretargeting Therapeutics in PSMA-Positive Prostate Cancer

Журнал:

Molecular Pharmaceutics

Рік:

2019

Файл:

PDF, 5.61 MB

2019

Structural and in Vivo Characterization of Tubastatin A, a Widely Used Histone Deacetylase 6 Inhibitor

Shen, Sida, Svoboda, Michal, Zhang, Guangming, Cavasin, Maria A, Motlova, Lucia, McKinsey, Timothy A, Eubanks, James H, Bařinka, Cyril, Kozikowski, Alan P

Журнал: